Iityhubhu zeLebhu

Imveliso

Ivermectin 70288-86-7 Anti-Parasitics Antibiotic

Inkcazelo emfutshane:

Izithethantonye:Ivermectine

Inombolo yeCAS:70288-86-7

Umgangatho:EP9

Ifomula yemolekyuli:C48H74O14

Ubunzima beFomula:875.09


Iinkcukacha zeMveliso

Iithegi zeMveliso

Intlawulo:T/T, L/C
Imvelaphi yeMveliso:eTshayina
Indawo yokuthumela ngenqanawa:Beijing/Shanghai/Hangzhou
Umthamo wemveliso:500kg/ngenyanga
Umyalelo(MOQ):25kg
Ixesha lokukhokhela:Iintsuku zokusebenza ezi-3
Imeko yokugcina:Igcinwe kwindawo epholileyo, eyomileyo, ubushushu begumbi.
Ipakethe imathiriyeli:igubu
Ubungakanani bepakethi:25kg/igubu
Ulwazi ngokhuseleko:UN2811 6.1/ PG 1

Ivermectin

Intshayelelo

I-Ivermectin iphuma kwi-Avermectin, sisibulali-zinambuzane esitsha esisebenzayo se-semisynthetic, i-acaricide kunye ne-nematicide, eye-arhente ye-nerve yezinambuzane kunye ne-biological penetrant.Inkqubo yesenzo kukuphazamisa imisebenzi ye-neurophysiological yezinambuzane kunye nokuvuselela ukukhululwa kwazo i-γ- i-aminobutyric acid isebenza kwi-nerve kunye ne-muscle junctions, yandisa ukukhululwa kwe-ion chloride, inqanda ukuhanjiswa kolwazi lwe-nerve junctions, kwaye ikhokelela ekukhubazekeni kunye nokufa okunetyhefu. yezinambuzane kunye namangolwane.Imveliso ayinambala okanye incindi emdaka etyheli.

Ivermectin, lichiza antiparasite.Okokuqala yayisetyenziswa kunyango lwezilwanyana ukunqanda kunye nokunyanga intshulube yentliziyo kunye ne-acariasis.

Ivermectin i-spectrum entsha ebanzi, eliphezulu-ukusebenza kunye netyhefu ephantsi antiparasitic ichiza, nto leyo enefuthe elihle lokugxotha kwizimfimfithi zangaphakathi nangaphandle, ingakumbi nematodes kunye arthropods.Kodwa ayinamsebenzi kwi-tapeworm, i-trematode kunye ne-protozoa.

Kule mihla, isetyenziselwa ukunyanga uhlaselo olubandakanya iintwala zentloko, ukhwekhwe, ubumfama bomlambo, i-strongyloidiasis, i-trichuriasis, i-ascariasis kunye ne-lymphatic filariasis.Isebenza ngeendlela ezininzi zokubulala i-parasites ekujoliswe kuyo, kwaye ingathathwa ngomlomo, okanye ifakwe esikhumbeni ngenxa yokuhlaselwa kwangaphandle.Yeyosapho lwe-avermectin yamayeza.

Ngumgubo wekristale omhlophe okanye omthubi, onyibilikayo kwi-methanol, ii-esters kunye neehydrocarbons ezinuka kamnandi, ezinganyibilikiyo emanzini.Iinaliti kunye neepilisi ezenziwe nge-ivermectin zisetyenziselwa ukunyanga i-nematodiasis yesisu, iimpethu ze-bovine fly, iimpethu ze-dermatoglyphic fly, iimpethu zempumlo zegusha, ihagu kunye nokhwekhwe lwegusha kwizilwanyana zasekhaya.Ngaphandle koko, i-Ivermectin ingasetyenziselwa ukunyanga i-nematodes ye-parasitic kwiinkukhu ezifana ne-Ascaris, i-pulmonary nematodes, njl. njl. ezizifunxi-gazi ngokubanzi kwizityalo.Iimpawu ezibalaseleyo ziziphumo ebezingalindelekanga zokukhanya, ukusetyenziswa kweziyobisi okwexesha elinye ngaxeshanye kunokubulala iintlobo ngeentlobo zezifunxi-gazi kwi-vivo nakwi-vitro zombini.

Inkcazo (EP9)

Into

Inkcazo

Imbonakalo I-crystalline powder emhlophe okanye etyheli-mhlophe
Ukunyibilika Ngokuqhelekileyo ayinyibiliki emanzini, i-soluble ngokukhululekileyo kwi-methylene chloride, i-soluble etywaleni.
Ukuchongwa I-IR: ihambelana naleyo yomgangatho we-CRS
I-HPLC: ixesha lokugcinwa kwe-H2B1a kunye ne-H2B1b ihambelana nelo lolungiselelo oluqhelekileyo
Ukubonakala kwesisombululo Icacile kwaye ayinambala kakhulu kune-BY7
Ukujikeleza okuthe ngqo (i-anhydours kunye ne-solvent-free substance) -17 ukuya -20 °

Izinto eziyeleleneyo (%)

Ukungcola komntu ngamnye (RRT1.3-1.5)≤2.5
Nakuphi na okunye ukungcola komntu≤1
Iyonke≤5
Ukungahoyi umda≤0.05
IEthanol kunye neformamide (%) I-Ethanol≤5.0
Formamide≤3.0
Amanzi (%) ≤1.0
Uthuthu olufakwe emanzini (%) ≤0.1
Ikati (ug/g) ≤1
Uvavanyo (%), (HPLC, isiseko sokumisa) H2B1A/(H2B1a + H2B1b) ≥ 90.0
95.0≤H2B1a + H2B1b≤102.0

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