Iityhubhu zeLebhu

Imveliso

I-Romifidine HCL 65896-14-2 iMetabolites

Inkcazelo emfutshane:

Izithethantonye:1H-Imidazol-2-amine, N-(2-bromo-6-fluorophenyl)-4,5-dihydro-, monohydrochloride

Inombolo yeCAS:65896-14-2

Umgangatho:endlwini

Ifomula yemolekyuli:I-C9H10BrClFN3

Ubunzima beFomula:294.55


Iinkcukacha zeMveliso

Iithegi zeMveliso

Intlawulo:T/T, L/C
Imvelaphi yeMveliso:eTshayina
Indawo yokuthumela ngenqanawa:Beijing/Shanghai/Hangzhou
Umthamo wemveliso:2kg/ngenyanga
Umyalelo(MOQ):10g
Ixesha lokukhokhela:Iintsuku zokusebenza ezi-3
Imeko yokugcina:Igcinwe kwindawo epholileyo, eyomileyo, ubushushu begumbi.
Ipakethe imathiriyeli:ingqayi
Ubungakanani bepakethi:10g/ibhodlela
Ulwazi ngokhuseleko:UN 2811 6.1/PG 3

I-Romifidine HCL

Intshayelelo

I-Romifidine liyeza elisetyenziswa kunyango lwezilwanyana njengento yokuthomalalisa ikakhulu kwizilwanyana ezinkulu ezifana namahashe, nangona inokusetyenziswa kwiindidi ezahlukeneyo zeentlobo.Ayisetyenziswa ebantwini, kodwa inxulumene ngokusondeleyo kwisakhiwo kwi-clonidine yeziyobisi ezisetyenziswa ngokuqhelekileyo.

I-Romifidine isebenza njenge-agonist kwi-α2 i-adrenergic receptor subtype.Imiphumo emibi ingabandakanya i-bradycardia kunye nokudandatheka kokuphefumula.Ihlala isetyenziswa kunye nezinye iziyobisi ezithomalalisa okanye ezidambisa iintlungu ezifana ne-ketamine okanye i-butorphanol.I-Yohimbine ingasetyenziselwa njenge-antidote yokuguqula ngokukhawuleza imiphumo.

Inkcazo (kwimigangatho yendlu)

Into

Inkcazo

Imbonakalo

Okumhlophe okuqinileyo

Ukunyibilika

Inyibilika kancinane kwi-DMSO, iMethanol naManzi

Indawo yokunyibilika

256 ~ 260℃

Ukuchongwa

NMR;LC-MS

Uvavanyo (HPLC)

98% min.


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