Iityhubhu zeLebhu

Imveliso

I-Oxytocin 50-56-6 IHormone kunye ne-endocrine Ukusetyenziswa komntu

Inkcazelo emfutshane:

Izithethantonye:(1-hemicystine) -oxytocin;i-di-sipidin;endopituitrina

Inombolo yeCAS:50-56-6

Umgangatho:USP41

Ifomula yemolekyuli:I-C43H66N12O12S2

Ubunzima beFomula:1007.19


Iinkcukacha zeMveliso

Iithegi zeMveliso

Intlawulo:T/T, L/C
Imvelaphi yeMveliso:eTshayina
Indawo yokuthumela ngenqanawa:Beijing/Shanghai/Hangzhou
Umthamo wemveliso:1kg/ngenyanga
Umyalelo(MOQ):10g
Ixesha lokukhokhela:Iintsuku zokusebenza ezi-3
Imeko yokugcina:I-2-8℃ yokugcina ixesha elide, ikhuselwe ekukhanyeni
Ipakethe imathiriyeli:ingqayi
Ubungakanani bepakethi:10g/ibhodlela
Ulwazi ngokhuseleko:Ayizompahla eziyingozi

Oxytocin

Intshayelelo

I-Oxytocin, i-hormone ye-peptide kunye ne-neuropeptide, uhlobo lweyeza le-uterine contractile, elinokukhutshwa kwi-pituitary yangasemva yezilwanyana okanye i-synthesized chemically.Ukuba zidityaniswe ngeekhemikhali ezingenayo i-vasopressin kwaye azinampembelelo yoxinzelelo.

Inokukhetha ngokukhetha i-uterine muscle egudileyo kwaye yomeleze ukucutheka kwayo.Isibeleko sesibeleko sinovelwano kakhulu kwi-oxytocin ngenxa yokunyuswa kokukhuselwa kwe-estrogen.Isibeleko esingekavuthwa asinakusabela kule mveliso.Impendulo yesibeleko kwi-oxytocin yayiphantsi kwithuba lokuqala okanye eliphakathi kwithuba leenyanga ezintathu zokukhulelwa, kodwa yanda ngokuthe ngcembe kwithuba lekota yokugqibela yokukhulelwa, yaza yafikelela kwelona nani liphezulu ngaphambi kokubeleka.

I-dose encinci inokomeleza ukucutshungulwa kwesingqisho se-muscle egudileyo ezantsi kwesibeleko, ukomeleza ukunyanzeliswa kwayo, ukukhawulezisa ukuphindaphinda kwe-contraction, kunye nokugcina i-polarity kunye ne-symmetry efana nokuhanjiswa kwendalo.Ke ngoko, isetyenziselwa uklinikhi ukwenza umsebenzi okanye i-oxytocia.

Idosi enkulu yenza isivumelwano semisipha ye-uterine ngendlela ye-tetanic.Isetyenziselwa uklinikhi ukucinezela imithambo yegazi phakathi kwemicu yezihlunu, ukuthintela ukopha kwangemva kokubeleka kunye nokungaphelelanga kokuphuma kwangemva kokubeleka.Ikhuthaza i-lactation, iyancipha i-mammary duct, kwaye ikhuthaza ukukhutshwa kobisi kwibele.Nangona kunjalo, ayikwazi ukunyusa ukukhutshwa kobisi, kodwa inokukhuthaza kuphela ukukhutshwa kobisi.

I-Oxytocin isoloko idityaniswa nokulungiswa kwe-ergot ukunyanga ukopha kwasemva kokubeleka.Isetyenziselwa ikakhulu ukuzala ngexesha lokukhulelwa kade kunye nokulibaziseka kokubeleka okubangelwa yi-atoni yesibeleko ngexesha lokubeleka.Ikwasetyenziselwa uvavanyo lwe-oxytocin sensitivity kunye nokunceda ekukhupheni ubisi lwasemva kokubeleka.

I-Oxytocin ikhutshelwa kumjikelezo wegazi njengehomoni ekuphenduleni umsebenzi wesondo kunye nangexesha lokubeleka.Ikwafumaneka nakwifomu yamayeza.Kuyo nayiphi na indlela, i-oxytocin ivuselela ukufinyela kwesibeleko ukukhawulezisa inkqubo yokuzala.Ukuveliswa kunye nokukhutshwa kwe-oxytocin kulawulwa yindlela efanelekileyo yokuphendula, apho ukukhutshwa kwayo kokuqala kukhuthaza ukuveliswa kunye nokukhululwa kwe-oxytocin eyongezelelweyo.

Inkcazo (USP41)

Into

Inkcazo

Imbonakalo Imhlophe okanye iphantse imhlophe, i-hygroscopic powder
Ukuchongwa I-HPLC: Ixesha lokugcinwa liyafana nereferensi
Ubunzima be-Ion yeMolekyuli: 1007.2
Umxholo we-amino acid

Asp: 0.95 ukuba 1.05

Glu: 0.95 ukuba 1.05

Gly: 0.95 ukuya 1.05

Pro: 0.95 ukuba 1.05

Tyr: 0.70 ukuba 1.05

Leu: 0.90 ukuba 1.10

Ile: 0.90 ukuba 1.10

Cys: 1.40 ukuba 2.10

Izinto ezinxulumeneyo Ubumdaka bubonke i-NMT 5%
Isiqulatho samanzi (KF) NMT 5.0%
Umxholo we-Acetic acid 6%-10%
Intsalela yezinyibilikisi (GC)
Acetonitrile NMT 410 ppm
I-methylene chloride NMT 600 ppm
Isopropylether NMT 4800 ppm
Ehtanol NMT 5000 ppm
N, N-Dimethyl Formanide NMT 880 ppm
Ubalo lweMicrobial NMT 200 cfu/g
Umsebenzi NLT 400 USP Oxytocin Units nge mg

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