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Ukusetyenziswa kweDoramectin kunyango lwezifo

Doramectin, luhlobo olutsha lweyeza elibanzi-spectrum antiparasitic ezayo fm usapho avermectin.Impembelelo ye-insecticidal ingcono kune-avermectin kunye ne-ivermectin.Lichiza lamva nje lonyango lwezilwanyana kwihlabathi.Ingasetyenziselwa ukunyanga kunye nokuthintela izifo ezibangelwa yi-nematodes kwi-gastrointestinal tract, imiphunga, ii-subcutaneous tissues kunye ne-lacrimal ducts yenkomo, iigusha kunye neehagu, kunye nezifo ezibangelwa yimpethu, ukhwekhwe, iintwala kunye namakhalane kwi-subcutaneous kunye ne-nasal tract. .

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1. Ukukhupha okanye ukubulala i-parasite

I-Doramectin inempembelelo ebanzi yokugxotha kwizilwanyana zangaphakathi nangaphandle, ngakumbi kwi-nematodes yesisu kunye ne-arthropods, kodwa ayinampembelelo kwi-tapeworms, i-trematodes kunye ne-protozoa.

Kuye kwaphuculwa ukuba izinga elisebenzayo le-Doramectin ngokuchasene nezigaba ezikhulileyo kunye nezingavuthwanga zeenkomo kunye neegusha, ezifana ne-Ostromella elegans, i-Kechen Ostromella, i-Haematostrongylus twister, i-Hemitis twister, i-Trichostrongylus ehrlii, i-Trichostrongylus serpentinus, i-Cupressus punctatus, i-Cupressus punctatus, ekwaziwa njenge hookworm), iTrichostrongylus papillaris kunye neRadiated Nodular Nematodes, yi-99%.

Izinga elisebenzayo ngokuchasene ne-Trichostrongylus spinosus yi-93% ~ 99%;

Ireyithi esebenzayo yeTrichuris yi-92.3% ~ 94.6%;

Umlinganiselo osebenzayo we-nematode Spoonae yi-96.5%;

Amazinga asebenzayo kubantu abadala kunye nemibungu ye-Nematodes helleri yi-73.3% kunye ne-75.5% ngokulandelanayo (ezinye iingxelo ziyi-97.9%);

Umlinganiselo osebenzayo wokufunxa i-nematode emehlweni eenkomo yi-100%.

I-Doramectin iyasebenza ngokuchasene neentlobo ezahlukeneyo ze-arthropod parasites ezinkomeni.

Izinga elisebenzayo lokulwa namantwala, ukhwekhwe, iintwala zegazi kunye neempukane zofele lwenkomo (inqanaba lokuqala, lesibini nelesithathu) ezifumaneka ngokwemvelo ezinkomeni yi-100%;

Izinga elisebenzayo lembungu, i-nodule worm (odontophagostomus nematode), i-pulmonary nematode (postroundworm), intshulube ebomvu kunye ne-blue pine nematode ezihagwini yi-100%;

Izinga elisebenzayo kwintwala yegazi yehagu kunye nokhwekhwe yi-100%.

2. Iimpawu ze-Pharmacodynamic

I-Doramectin kulula ukufunxwa kwindawo yokutofa, i-bioavailability ye-subcutaneous kunye ne-intramuscular injection iphantse ifane, kwaye naliti ayinalo uxinzelelo kunye neentlungu.Inomphumo omude kunye osebenzayo kwaye unokugcina ugxininiso lonyango egazini lezilwanyana ixesha elide, ngoko ke ixesha lokukhusela lide.I-Doramectin ineziphumo ebezingalindelekanga ezincinci kwaye ingasetyenziswa zizilwanyana ezincinci.Ayinayo i-carcinogenic, i-teratogenic kunye nemiphumo ye-mutagenic, akukho mpembelelo kwi-immunity emva kokugonywa.

Uphononongo lwakutsha nje luqinisekisile ukuba iintsalela ze-doramectin ezikhutshiweyo ngeelindle zisagcina ukusebenza kokubulala izinambuzane, kodwa kuxhomekeke kwiimpawu ezibonakalayo zelindle kunye nokutshintsha kweemeko zemozulu.

Thina i-Xiamen Neore singabathengisi bokwenza i-API abanamava angaphezulu kweminyaka eli-15 kushishino lwamayeza e-China.Sibonelela ngeDoramectin ngomgangatho ophezulu kunye nexabiso elikhuphisanayo.

Wamkelekile ngokufudumeleyo cela ikowuti.

Sikwimeko entle ukuba singakuboneleli kuphela ngemathiriyeli ekrwada ekumgangatho ophezulu, kodwa kunye neyona nto ibalaseleyo ekuboneleleni phambi/ emva kwenkonzo yokuthengisa.Iqela lethu le-R&D liya kukunika nayiphi na inkxaso yobugcisa.


Ixesha lokuposa: Feb-21-2023