Iityhubhu zeLebhu

Imveliso

Doramectin 117704-25-3 Anti-Parasitics Antibiotic

Inkcazelo emfutshane:

Izithethantonye:25-Cclohexyl-avermectin B1, Avermectin A1a

Inombolo yeCAS:117704-25-3

Umgangatho:endlwini

Ifomula yemolekyuli:C50H74O14

Ubunzima beFomula:899.11


Iinkcukacha zeMveliso

Iithegi zeMveliso

Intlawulo:T/T, L/C
Imvelaphi yeMveliso:eTshayina
Indawo yokuthumela ngenqanawa:Beijing/Shanghai/Hangzhou
Umthamo wemveliso:15kg/ngenyanga
Umyalelo(MOQ):1kg
Ixesha lokukhokhela:Iintsuku zokusebenza ezi-3
Imeko yokugcina:Gcina kwiqondo lobushushu 2-8℃ ixesha elide, ukhuselwe ekukhanyeni.
Ipakethe imathiriyeli:ibhotile
Ubungakanani bepakethi:1kg/igubu
Ulwazi ngokhuseleko:UN 2811 6.1/ PG 3

Doramectin

Intshayelelo

I-Dorametin liyeza elitsha le-macrolide antiparasite.Sisithinteli-ntsholongwane se-avermectin esiveliswe ngokubiliswa kohlobo olutsha lwe-Streptomyces avermitis ene-cyclohexamic acid njenge-precursor.Kuthathwa njengelinye lawona machiza alungileyo e-antiparasite kusapho lwe-avermectin.

Impembelelo ye-insect ye-insect ye-Doramectin ifana ne-Ivermectin, enokuthintela ukuhanjiswa kweentsholongwane ze-nerve phakathi kwee-nerve kunye nezihlunu, kwaye yenza inambuzane ikhubazekile kwaye ife kude nomkhosi.Nangona kunjalo, ngenxa yoxinaniso lwegazi oluphezulu lwe-doramectin emzimbeni, ukupheliswa kukucotha kakhulu, kwaye ixesha lokugcinwa kokusebenza lide, ngoko ke umphumo wokugxotha inambuzane ungcono kune-Ivermectin.Ngenxa yokuba akukho kusabela komzimba xa usebenzisa i-Doramectin, ngoko kukhuseleko olungakumbi olunokusetyenziswa.Ikwathathwa njengechiza endaweni ye-Ivermectin.

Isetyenziselwa unyango kunye nolawulo lwe-parasitosis yangaphakathi (i-nematodes yesisu kunye ne-pulmonary), amakhalane kunye ne-mange (kunye nezinye i-ectoparasites).

Ngokwekliniki ibonisa ukuba iDoramectin inefuthe elihle kwi-nematodes kwindlela yokwetyisa yeehagu.Ngokutsho kwengxelo, iihagu zilawulwa nge-intramuscularly kwi-dose ye-0.3 mg / kg ubunzima bomzimba.Inzuzo yobunzima bosulelo olwenziweyo kunye namatyala osulelo lwendalo lwaluphezulu kakhulu kunelo qela lolawulo kwi-7, 14 kunye ne-21 iintsuku emva kokulawulwa.Xa kuthelekiswa neqela lolawulo, iimbungu zisuswe nge-100% ngaphandle kwemiphumo emibi.

Ikwabonisa ngokweklinikhi kunyango lweSarcoptes ukhwekhwe, kukho iziphumo ezilungileyo ukusuka kumantshontsho amantshontsho ancancayo ukuya kwiimazi.

I-Doramectin iyafumaneka kumahashe njengomlomo, i-flavored, ijeli ye-bioadhesive phantsi kwegama.

I-Doramectin ayizinzile kwindalo.Ibola ngokukhawuleza kwaye ayisebenzi phantsi kokukhanya kwelanga.Amachiza ayo ashiyekileyo ayityhefu kwiintlanzi nakwizinto eziphila emanzini.Ngoko ke, kufuneka kuqwalaselwe ingqalelo ekukhuselweni komthombo wamanzi.

Inkcazo (kwiMgangatho weNdlu)

Into

Inkcazo

Imbonakalo Umgubo omhlophe wekristale
Ukuchongwa HPLC, IR
Ukubonakala kwesisombululo Isisombululo sicacile kwaye asinambala kakhulu kunesisombululo sereferensi BY6
Amanzi ≤3%
Intsimbi enzima ≤20ppm
Uthuthu lweSulfate ≤0.1%
BHT ≤2000ppm
Into enxulumeneyo IAvermectin B1a≤1.5%
IAvermectin B1b≤1.0%
IAvermectin B1a kunye neAvermectin B1b≤2.0%
Ubumdaka bubonke i-NMT 5.0%
Isinyibilikisi esishiyekileyo I-acetone≤5000ppm
I-Ethanol≤30000ppm
I-Ethyl acetate≤5000ppm
Methanol≤3000ppm
Isivavanyi ≥95% (kwisiseko se-anhydrous kunye ne-solvent free)

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