Iityhubhu zeLebhu

Imveliso

I-Oclacitinib maleate 1208319-27-0 Anti-inflammatory NSAID

Inkcazelo emfutshane:

Igama lemveliso:Oclacitinib maleate
Izithethantonye:Oclacitinib PF-03394197
Inombolo yeCAS:1208319-27-0
Umgangatho:endlwini
Ifomula yemolekyuli:I-C19H27N5O6S
Ubunzima bemolekyuli:453.51


Iinkcukacha zeMveliso

Iithegi zeMveliso

Intlawulo:T/T, L/C
Imvelaphi yeMveliso:eTshayina
Indawo yokuthumela ngenqanawa:Beijing/Shanghai/Hangzhou
Iodolo (MOQ):10g
Ixesha lokukhokhela:3 iintsuku zokusebenza
Umthamo wemveliso:5kg/ngenyanga
Imeko yokugcina:Igcinwe kwindawo epholileyo, eyomileyo, ubushushu begumbi.
Ipakethe imathiriyeli:ingqayi
Ubungakanani bepakethi:10g/ibhodlela
Ulwazi ngokhuseleko:Ayizompahla eziyingozi

Oclacitinib maleate

Intshayelelo

I-Oclacitinib, iyeza lonyango lwezilwanyana elisetyenziselwa ukulawula i-atopic dermatitis kunye ne-pruritus evela kwi-allergic dermatitis kwizinja ubuncinane kwiinyanga ezili-12 ubudala.I-Chemical, i-synthetic cyclohexylamino pyrrolopyrimidine janus kinase inhibitor ekhethiweyo ngokufanelekileyo kwi-JAK1.Ivimbela ukuhanjiswa kwesignali xa i-JAK ivuliwe kwaye ngaloo ndlela inceda ukunciphisa ukubonakaliswa kwee-cytokines ezivuthayo.

I-Oclacitinib ibhalwe ukunyanga i-atopic dermatitis kunye nokurhawuzelela (i-pruritus) okubangelwa kukwaliwa kwizinja, nangona ikwasetyenziselwe ukunciphisa ukurhawuzelela kunye ne-dermatitis ebangelwa ziinfestations zentakumba.Ithathwa njengesebenza kakhulu kwizinja, kwaye iye yasekwa njengekhuselekile ukusetyenziswa kwexesha elifutshane.

Inkcazo (kwimigangatho yendlu)

Into

Inkcazo

Imbonakalo Okumhlophe okuqinileyo
HNMR Ukuthobela isakhiwo
I-LC-MS Ukuthobela isakhiwo
Ubunyulu ≥98%
Indawo yokunyibilika N / A

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