Iityhubhu zeLebhu

Imveliso

Mirabegron 223673-61-8 Inhibitor Umqondiso we-Neuronal

Inkcazelo emfutshane:

Izithethantonye:YM 178,N-(4-(2-(2-hydroxy-2-phenylethylamino)ethyl)phenyl)-2-(2-aminothiazol-4-yl)acetamide

Inombolo yeCAS:223673-61-8

Umgangatho:endlwini

Ifomula yemolekyuli:I-C21H24N4O2S

Ubunzima beFomula:396.51


Iinkcukacha zeMveliso

Iithegi zeMveliso

Intlawulo:T/T, L/C
Imvelaphi yeMveliso:eTshayina
Indawo yokuthumela ngenqanawa:Beijing/Shanghai/Hangzhou
Umthamo wemveliso:100kg/ngenyanga
Umyalelo(MOQ):25kg
Ixesha lokukhokhela:Iintsuku zokusebenza ezi-3
Imeko yokugcina:Igcinwe kwindawo epholileyo, eyomileyo, ubushushu begumbi.
Ipakethe imathiriyeli:igubu
Ubungakanani bepakethi:25kg/igubu
Ulwazi ngokhuseleko:Ayizompahla eziyingozi

I-Mirabegron

Intshayelelo

I-Mirabegron, i-beta-3 i-adrenergic receptor agonist, evuselela i-beta-3 adrenergic receptor kwaye iphumle i-detrusor muscle egudileyo, ngaloo ndlela ikhulise umthamo wesinye kwaye isetyenziselwa ukunyanga iimpawu ze-bladder esebenzayo (OAB), ezifana nokukhawuleza ukungazinzi, ukukhawuleza, kunye namaxesha.

Izibonelelo zayo zifana neyeza le-antimuscarinic ezifana ne-solifenacin okanye i-tolterodine.

Inkcazo (USP/EP)

Into

Inkcazo

Imbonakalo Mhlophe ukuya kumgubo omhlophe

Ukuchongwa

IR, HPLC
Isiqulatho samanzi NMT 0.5%
Intsalela ekutshisweni NMT 0.1%
Intsimbi enzima NMT 20ppm
Umxholo wePalladium NMT 20ppm
Isomer ye-Optical NTM 0.5%
Into enxulumeneyo Z-168*: NMT 0.15%
  SC03610*: NMT 0.15%
  Nakuphi na okunye ukungcola okungaziwayo: NMT 0.10%
  Ukungacoceki kukonke: NMT 0.5%
I-2-(2-aminothianzol-4-yl) i-acetic acid NMT 0.1%
Isinyibilikisi esishiyekileyo IMethanol: NMT 0.3%
  I-Ethyl acetate: NMT 0.5%
  THF: NMT 0.072%
  I-Benzene: NMT 0.0002%
  Itoluene: NMT 0.089%
Isivavanyi 98.0% - 102.0%
PSD D (0.5): 10μm - 30μm
  D (0.9): 20μm - 80μm

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