Iityhubhu zeLebhu

Imveliso

I-Detomidine HCl 90038-01-0 Inhibitor Neuronal signal Analgesic

Inkcazelo emfutshane:

Izithethantonye:I-Detomidine hydrochloride, 5-(2,3-Dimethylbenzyl) imidazole Hydrochloride

Inombolo yeCAS:90038-01-0

Umgangatho:endlwini

Ifomula yemolekyuli:I-C12H15ClN2

Ubunzima beFomula:222.71


Iinkcukacha zeMveliso

Iithegi zeMveliso

Intlawulo:T/T, L/C
Imvelaphi yeMveliso:eTshayina
Indawo yokuthumela ngenqanawa:Beijing/Shanghai/Hangzhou
Umthamo wemveliso:50kg/ngenyanga
Umyalelo(MOQ):25kg
Ixesha lokukhokhela:Iintsuku zokusebenza ezi-3
Imeko yokugcina:Igcinwe kwindawo epholileyo neyomileyo, ivalwe kwaye igcinwe kude nokukhanya.
Ipakethe imathiriyeli:igubu
Ubungakanani bepakethi:25kg/igubu
Ulwazi ngokhuseleko:Ayizompahla eziyingozi

I-Detomidine HCl

Intshayelelo

I-Detomidine i-imidazole derivative kunye ne-α2-adrenergic agonist, isetyenziswe njengesilwanyana esikhulu sezilwanyana, esisetyenziswa ngokukodwa kumahashe.

I-Detomidine i-sedative eneempawu ze-analgesic i-α2-adrenergic agonists ivelisa i-dose-dependent sedative kunye ne-analgesic effects, i-mediated by activation ye-α2 catecholamine receptors, ngaloo ndlela ibangela impendulo engalunganga, ukunciphisa ukuveliswa kwee-neurotransmitters ezinomdla.

Inkcazo (kwimigangatho yendlu)

Into

Inkcazo

Imbonakalo

Ikristale emhlophe okanye ephantse ibe mhlophe okanye umgubo

Ukunyibilika

Inyibilika emanzini, i-methanol kunye ne-DMSO

Indawo yokunyibilika

158℃~162℃

Ukuchongwa

NMR

Ukungcola okukodwa okukhulu

≤0.2%

Ukungcola ngokupheleleyo

≤1.0%

Amanzi (KF)

≤1.0%

Intsalela ekutshisweni

≤0.10%

I-acetone

≤0.5%

IMethanol

≤0.3%

I-Ethyl acetate

≤0.5%

Tetrahydrofuran

≤0.072%

Isivavanyi Iqulethe 98.0% -102.0% yeC12H14N2.HCl(Kwisiseko se-anhydrous)

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  • Okulandelayo: